Prof. Debabrata Maiti is an Indian scientist specializing in organometallic chemistry and bioinspired catalysis and serving as a Professor of Chemistry at the Indian Institute of Technology Bombay, Mumbai. He was awarded the Shanti Swarup Bhatnagar Prize, the prestigious Indian national award for excellence in scientific research, for Chemical Sciences for the year 2022 for his significant contributions to developing transition metal catalysis for transforming organic molecules to prepare value-added materials by site- selective functionalization, leading impact on agrochemicals and pharmaceuticals industry.
Day 1 - Session Details
MODULE – 1 : C-H activation: 1 & 2
Concepts Covered:
Initial idea about C-H activation
N-Heterocycle synthesis through C–H activation /annulation cascade
Learning Outcomes
Students get a first idea of C-H activation and N heterocycle synthesis through the C-H activation/annulation cascade.
MODULE – 2 : C-H activation: 3 & 4
Concepts Covered:
C–H arylation for drug scaffolds
C–H borylation /silylation in medicinal chemistry
Learning Outcomes
Students get a first idea of C–H arylation for drug scaffolds and C–H borylation /silylation in medicinal chemistry.
MODULE – 3 : C-H activation: 5 & 6
Concepts Covered:
C–H amination in drug discovery
C–H fluorination /fluoroalkylation in drug discovery
Learning Outcomes
Students get a first idea of C–H amination in drug discovery and C–H fluorination /fluoroalkylation in drug discovery.
MODULE – 4 : C-H activation: 7 & 8
Concepts Covered:
C–H methylation: the methyl magic presumed in drug discovery
Amino acid, peptide and protein modification through C–H activation
Learning Outcomes :
Students get a first idea of C–H methylation: the methyl magic presumed in drug discovery and amino acid, peptide, and protein modification through C–H activation.
Day 2 - Session Details
MODULE – 5 : C-H activation: 9 & 10
Concepts Covered:
Bioimaging/ radiolabelling via C–H activation
Bioconjugation through C–H activation
Learning Outcomes
Students get an introduction to bioimaging/radiolabelling via C–H activation and bioconjugation through C–H activation.
MODULE – 6 : C-H activation: 11 & 12
Concepts Covered:
Drug-metabolite synthesis through C–H oxidation
Late-stage C–H functionalization of drug molecules
Learning Outcomes
Students understand drug-metabolite synthesis through C–H oxidation and late-stage C–H functionalization of drug molecules.
MODULE – 7 : C-H activation: 13 & 14
Concepts Covered:
DNA-encoded library development through C–H activation
Case studies of drug/drug-like molecule synthesis via C–H activation
Learning Outcomes
Students learn about DNA-encoded library development through C–H activation and case studies of drug/drug-like molecule synthesis via C–H activation.
MODULE – 8 : C-H activation: 15
Concepts Covered:
Summary of C-H activation methodology
Learning Outcomes:
Students understand the importance of C–H activation methodologies and their benefits to mankind.
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